SCHEMBL4603045

SCHEMBL4603045

CCCOc1ccc(-c2cc(F)cc(C(=O)O)c2)cc1C(=O)NC(CO)Cc1c[nH]c2ccc(F)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 2/20 0.40
ICAM1 P05362 2/20 0.40
ITGAL P20701 2/20 0.40
PPARG P37231 2/20 0.39
CCKBR P32239 2/20 0.38
HTR2A P28223 2/20 0.38
HTR1A P08908 2/20 0.38
TSHR P16473 1/20 0.37
SCN8A Q9UQD0 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
PTPN11 Q06124 1/20 0.37
HTT P42858 1/20 0.37
HTR2C P28335 1/20 0.37
SLC6A4 P31645 1/20 0.37
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
ADAM17 P78536 1/20 0.36
TRPV1 Q8NER1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14557691 0.94 HTR2A (0.40) ITGB2ICAM1ITGALPPARGCCKBR
SCHEMBL14557754 0.94 MPO (0.39) ITGB2ICAM1ITGALPPARGCCKBR
SCHEMBL4602963 0.94 PTPN11 (0.43) ITGB2ICAM1ITGALPPARGCCKBR
SCHEMBL4601908 0.92 ITGB2 (0.49) ITGB2ICAM1ITGALPPARGCCKBR
SCHEMBL14557733 0.92 HTR1A (0.38) ITGB2ICAM1ITGALPPARGCCKBR
SCHEMBL14557732 0.90 ICMT (0.39) ITGB2ICAM1ITGALPPARGCCKBR
SCHEMBL14557731 0.90 NR3C1 (0.40) ITGB2ICAM1ITGALCCKBRHTR2A
SCHEMBL14557960 0.89 PPARG (0.42) ITGB2ICAM1ITGALPPARGCCKBR
SCHEMBL14557719 0.89 ITGB2 (0.39) ITGB2ICAM1ITGALPPARGCCKBR
SCHEMBL14557962 0.89 ITGB2 (0.45) ITGB2ICAM1ITGALPPARGCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912970-A2 ACYLTRYPTOPHANOLS FOR FERTILITY CONTROL Bayer Schering Pharma Aktiengesellschaft (DE) 2008-04-23 EP disclosed
WO-2007017289-A2 ACYLTRYPTOPHANOLS FOR FERTILITY CONTROL BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-02-15 WO disclosed