SCHEMBL4602585

SCHEMBL4602585

N#Cc1cc(C#N)cc(Oc2ccc(CC(=O)Nc3ccc(S(N)(=O)=O)cc3Br)cc2Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 19/20 0.58
CA2 P00918 19/20 0.58
CA12 O43570 11/20 0.58
CA9 Q16790 11/20 0.58
CA5A P35218 3/20 0.53
CA7 P43166 3/20 0.53
CA5B Q9Y2D0 3/20 0.53
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4604104 0.90 CA2 (0.59) CA1CA2CA12CA9CA5A
SCHEMBL4603625 0.89 CA1 (0.58) CA1CA2CA12CA9CA5A
SCHEMBL4604312 0.87 CA1 (0.54) CA1CA2CA12CA9CA5A
SCHEMBL4604199 0.87 CA2 (0.58) CA1CA2CA12CA9CA5A
SCHEMBL4603727 0.86 CA1 (0.49) CA1CA2CA12CA9CA5A
SCHEMBL4604203 0.85 CA1 (0.56) CA1CA2CA12CA9CA5A
SCHEMBL4603542 0.85 MEN1 (0.53) MEN1KMT2A
SCHEMBL2638748 0.83 CA1 (0.59) CA1CA2CA12CA9CA5A
SCHEMBL4604671 0.83 CA1 (0.53) CA1CA2CA12CA9CA5A
SCHEMBL4603722 0.82 CA1 (0.49) CA1CA2CA12CA9CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940781-A1 PHENYL-ACETAMIDE NNRT INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2008-07-09 EP claimed
WO-2007045573-A1 PHENYL-ACETAMIDE NNRT INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2007-04-26 WO claimed