SCHEMBL4603530

SCHEMBL4603530

O=C(Br)NN1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.45
LIPE Q05469 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
TP53 P04637 1/20 0.37
GLA P06280 1/20 0.37
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
ALOX12 P18054 1/20 0.37
NFKB1 P19838 1/20 0.37
CNR1 P21554 2/20 0.34
CNR2 P34972 2/20 0.33
CA12 O43570 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7749096 0.79 HTT (0.45) HTTLIPEL3MBTL1LMNAPOLB
SCHEMBL7747487 0.79 HTT (0.45) HTTLIPEL3MBTL1LMNAPOLB
SCHEMBL1259794 0.79 HTT (0.45) HTTLIPEL3MBTL1LMNAPOLB
SCHEMBL15282042 0.79 HTT (0.45) HTTLIPEL3MBTL1LMNAPOLB
SCHEMBL7749230 0.79 HTT (0.45) HTTLIPEL3MBTL1LMNAPOLB
SCHEMBL21798768 0.78 HTT (0.48) HTTLIPEL3MBTL1LMNAPOLB
Hydrochloric Acid SCHEMBL27317890 0.77 HTT (0.44) HTTLIPEL3MBTL1LMNAPOLB
Hydrochloric Acid SCHEMBL27543811 0.77 HTT (0.44) HTTLIPEL3MBTL1LMNAPOLB
SCHEMBL244127 0.76
SCHEMBL3158910 0.76 HTT (0.47) HTTLIPEL3MBTL1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188290-B2 Reacting secondary amine, carbon dioxide, triarylsilyl chloride and halogenation agent GLAXO GROUP LIMITED (GB) 2012-05-29 US disclosed
US-20080262234-A1 Process for Preparing N, N-Substituted Carbamoyl Halides GLAXO GROUP LIMITED 2008-10-23 US disclosed
EP-1940783-A1 PROCESS FOR PREPARING N, N-SUBSTITUTED CARBAMOYL HALIDES GLAXO GROUP LIMITED (GB) 2008-07-09 EP disclosed
WO-2007048642-A1 PROCESS FOR PREPARING N, N-SUBSTITUTED CARBAMOYL HALIDES GLAXO GROUP LIMITED (GB) 2007-05-03 WO disclosed
WO-1995021155-A1 PROCESS FOR PREPARING N,N-SUBSTITUTED CARBAMOYL HALIDES FROM SECONDARY AMINES, CARBON DIOXIDE AND HALIDE-CONTAINING ELECTROPHILIC COMPOUNDS MONSANTO COMPANY (US) 1995-08-10 WO disclosed
US-5380855-A Carbon dioxide and secondary amine MONSANTO COMPANY (US) 1995-01-10 US disclosed