SCHEMBL4603963

SCHEMBL4603963

FC(F)(F)c1cccc(N2CCC(C(F)(F)F)CC2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.50
LCAT P04180 2/20 0.47
GRIN2B Q13224 3/20 0.47
DPP4 P27487 1/20 0.45
DPP9 Q86TI2 1/20 0.45
DPP7 Q9UHL4 1/20 0.45
DRD2 P14416 2/20 0.44
DRD3 P35462 2/20 0.44
ACACB O00763 4/20 0.43
CXCR3 P49682 1/20 0.43
PHGDH O43175 2/20 0.43
HTR1A P08908 1/20 0.43
HTR3E A5X5Y0 1/20 0.42
MEN1 O00255 1/20 0.42
HTR3B O95264 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30582911 0.87 HRH3 (0.52) HRH3LCATGRIN2BDPP4DPP9
SCHEMBL1351805 0.84 HTR3E (0.60) HRH3LCATGRIN2BDPP4DPP9
Hydrochloric Acid SCHEMBL5220893 0.83 HTR3E (0.59) HRH3LCATGRIN2BDPP4DPP9
SCHEMBL13059660 0.82 PRKCQ (0.54) HRH3LCATGRIN2BDPP4DPP9
SCHEMBL17667869 0.82 GRIN2B (0.49) HRH3LCATGRIN2BDPP4DPP9
SCHEMBL15918310 0.82 GRIN2B (0.49) HRH3LCATGRIN2BDRD2DRD3
SCHEMBL17062040 0.81 HRH3 (0.50) HRH3LCATGRIN2BDPP4DPP9
SCHEMBL31497599 0.81 HRH3 (0.50) HRH3LCATGRIN2BDPP4DPP9
SCHEMBL31497592 0.81 HRH3 (0.50) HRH3LCATGRIN2BDPP4DPP9
SCHEMBL22668979 0.80 GRIN2B (0.48) HRH3GRIN2BDRD2DRD3PHGDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940821-A2 NOVEL VANILLOID RECEPTOR LIGANDS AND THEIR USE FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2008-07-09 EP disclosed
WO-2007045462-A2 NOVEL VANILLOID RECEPTOR LIGANDS AND THEIR USE FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2007-04-26 WO disclosed