SCHEMBL4604581

SCHEMBL4604581

CC(Oc1ccc(OCc2cc(-c3ccc(C(F)(F)F)cc3)cc(-c3ccc(C(F)(F)F)cc3)c2)cc1)C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 10/20 0.69
PPARA Q07869 3/20 0.69
PPARG P37231 1/20 0.67
ADAMTS4 O75173 1/20 0.53
MMP13 P45452 1/20 0.53
FFAR1 O14842 4/20 0.53
PSEN1 P49768 2/20 0.51
PSEN2 P49810 2/20 0.51
APH1B Q8WW43 2/20 0.51
NCSTN Q92542 2/20 0.51
APH1A Q96BI3 2/20 0.51
PSENEN Q9NZ42 2/20 0.51
CYP1A2 P05177 1/20 0.50
GAA P10253 1/20 0.50
CYP2C9 P11712 1/20 0.50
PKM P14618 1/20 0.50
CYP2C19 P33261 1/20 0.50
MRGPRX4 Q96LA9 1/20 0.49
MAOB P27338 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21991483 0.88 MAOB (0.63) PPARAPPARGADAMTS4MMP13FFAR1
SCHEMBL25212758 0.81 CYP1A2 (0.59) PPARDPPARAPPARGCYP1A2GAA
SCHEMBL21057241 0.81 CYP1A2 (0.59) PPARDPPARAPPARGCYP1A2GAA
SCHEMBL11597291 0.81 CYP1A2 (0.59) PPARDPPARAPPARGCYP1A2GAA
SCHEMBL10946026 0.77 CYP1A2 (0.51) PPARDPPARAPPARGCYP1A2GAA
SCHEMBL8089170 0.77 CYP1A2 (0.54) PPARDPPARAPPARGCYP1A2GAA
SCHEMBL136831 0.77 CYP1A2 (0.54) PPARDPPARAPPARGCYP1A2GAA
SCHEMBL8089167 0.77 CYP1A2 (0.54) PPARDPPARAPPARGCYP1A2GAA
SCHEMBL11355228 0.77 CYP1A2 (0.49) PPARDPPARAMMP13PSEN1PSEN2
SCHEMBL1744700 0.77 CYP1A2 (0.64) PPARDPPARAPPARGFFAR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756062-A4 COMPOUNDS AND COMPOSITIONS AS PPAR MODULATORS IRM LLC (BM) 2008-01-02 EP disclosed
EP-1756062-A1 COMPOUNDS AND COMPOSITIONS AS PPAR MODULATORS IRM LLC (BM) 2007-02-28 EP disclosed
WO-2005113506-A1 COMPOUNDS AND COMPOSITIONS AS PPAR MODULATORS IRM LLC (BM) 2005-12-01 WO disclosed