SCHEMBL460537

SCHEMBL460537

C=CC/C=C(/N=C=O)C(=O)O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10818037 0.82
SCHEMBL10503949 0.75 GRIK1 (0.33)
SCHEMBL447238 0.75 GRIK1 (0.33)
SCHEMBL449264 0.72 GRIK1 (0.37)
SCHEMBL11432309 0.69
SCHEMBL451418 0.69 EP300 (0.44)
SCHEMBL3220907 0.69
SCHEMBL445701 0.68 EP300 (0.52)
SCHEMBL11879814 0.67
SCHEMBL27711431 0.67 KDM4E (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 70 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3898871-A1 COMPOSITION MADE FROM EPOXY RESIN AND POLYURETHANE Bostik SA (FR) 2021-10-27 EP claimed
WO-2020128326-A1 COMPOSITION MADE FROM EPOXY RESIN AND POLYURETHANE BOSTIK SA (FR) 2020-06-25 WO claimed
EP-2139938-B1 POLYMER POLYOL AND STABILIZER SYSTEMS BAYER ANTWERPEN NV (BE) 2011-12-21 EP claimed
EP-2139938-A1 POLYMER POLYOL AND STABILIZER SYSTEMS BAYER AG (DE) 2010-01-06 EP claimed
US-7064174-B2 Silicon containing compounds BIOCOMPATIBLES UK LIMITED (GB) 2006-06-20 US claimed
EP-1255761-B1 SILICON CONTAINING COMPOUNDS FROM MICHAEL - TYPE ADDITION REACTIONS USEFUL AS MONOMERS AND MACROMERS BIOCOMPATIBLES UK LTD (GB) 2005-08-31 EP claimed
EP-1122258-B1 Silicon containing compounds from Michael-type adduct reactions useful as monomers and macromers BIOCOMPATIBLES UK LTD (GB) 2004-05-12 EP claimed
US-20030152786-A1 Silicon containing compounds from michael-type addition reactions useful as monomers and macromers BIOCOMPATIBLES UK LIMITED (GB) 2003-08-14 US claimed
JP-2003522227-A 2003-07-22 JP claimed
EP-1255761-A1 SILICON CONTAINING COMPOUNDS FROM MICHAEL - TYPE ADDITION REACTIONS USEFUL AS MONOMERS AND MACROMERS BIOCOMPATIBLES LTD. (GB) 2002-11-13 EP claimed
WO-2001057048-A1 SILICON CONTAINING COMPOUNDS FROM MICHAEL - TYPE ADDITION REACTIONS USEFUL AS MONOMERS AND MACROMERS BIOCOMPATIBLES LIMITED (GB) 2001-08-09 WO claimed
EP-1122258-A1 Silicon containing compounds from Michael-type adduct reactions useful as monomers and macromers BIOCOMPATIBLES LIMITED (GB) 2001-08-08 EP claimed
US-6013731-A STABILIZER PRECURSOR BASED ON POLYOXYALKYLENE GLYCOL WITH LOW INDUCED UNSATURATION; IN SITU POLYMERIZATION OF VINYL MONOMERS AND POLYOLS TO FORM POLYMER POLYOLS OF HIGHER SOLIDS, LOWER VISCOSITY AND IMPROVED FILTERABILITY ARCO CHEMICAL TECHNOLOGY L.P. (US) 2000-01-11 US claimed
WO-1999031160-A1 POLYMER POLYOL AND STABILIZER SYSTEMS BAYER AG (DE) 1999-06-24 WO claimed
US-4822829-A Radiation-curable macromers based on (meth)acrylate-functional polyesters, and their use HUELS TROISDORF AKTIENGESELLSCHAFT (DE) 1989-04-18 US claimed
US-4820745-A SOLVENT-FREE HUELS TROISDORF AKTIENGESELLSCHAFT (DE) 1989-04-11 US claimed
US-11912801-B2 (Meth)acrylate urethane (urea) phosphonates as adhesion promoters 3M INNOVATIVE PROPERTIES COMPANY (US) 2024-02-27 US disclosed
EP-3898871-A1 COMPOSITION MADE FROM EPOXY RESIN AND POLYURETHANE Bostik SA (FR) 2021-10-27 EP disclosed
US-4304923-A REACTION PRODUCT OF POLYOL, POLYISOCYANATE, DICARBOXYLIC ACID, UNSATURATED COMPOUND MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1981-12-08 US disclosed
US-4228232-A NONSTICKING LITHOGRAPHIC PRINTING PLATES MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1980-10-14 US disclosed