SCHEMBL4607184

SCHEMBL4607184

O=C(O)N[C@H](CO)CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.51
CTSG P08311 1/20 0.50
CTRB1 P17538 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
HTT P42858 1/20 0.49
HPGD P15428 1/20 0.49
CYP3A4 P08684 1/20 0.47
MAPK1 P28482 1/20 0.47
TSHR P16473 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
POLB P06746 2/20 0.43
USP2 O75604 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3066768 1.00 CNR2 (0.51) CNR2CTSGCTRB1SMN1; SMN2KMT2A
SCHEMBL23201144 1.00 CNR2 (0.51) CNR2CTSGCTRB1SMN1; SMN2KMT2A
SCHEMBL4906710 0.87 TRPA1 (0.49)
SCHEMBL15958711 0.86 SMN1; SMN2 (0.50) CNR2CTSGCTRB1SMN1; SMN2KMT2A
SCHEMBL1177054 0.83 HTT (0.51) CNR2CTSGCTRB1SMN1; SMN2KMT2A
SCHEMBL3959317 0.81 MAPK1 (0.68) CTRB1KMT2AMEN1CYP3A4MAPK1
SCHEMBL3897966 0.81 MAPK1 (0.68) CTRB1KMT2AMEN1CYP3A4MAPK1
SCHEMBL2973301 0.81 MAPK1 (0.68) CTRB1KMT2AMEN1CYP3A4MAPK1
SCHEMBL23120332 0.81 SMN1; SMN2 (0.49) CNR2CTSGCTRB1SMN1; SMN2KMT2A
SCHEMBL14350867 0.81 SMN1; SMN2 (0.49) CNR2CTSGCTRB1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101466678-B Substituted 3-cyanopyridines as protein kinase inhibitors WYETH CORP 2012-12-26 CN disclosed
EP-1874768-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113837-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed