SCHEMBL4608516

SCHEMBL4608516

CN(Cc1ccc(C(=O)N2CC3CCC(CC3)C2)cc1)C(=O)c1cccc(C#N)c1.CN(Cc1ccc(C(=O)N2CC3CCC(CC3)C2)cc1)C(=O)c1cccc(F)c1.CN(Cc1ccc(C(=O)N2CC3CCC(CC3)C2)cc1)C(=O)c1ccccc1.CN(Cc1ccc(C(=O)N2CCCC3CCCCC32)cc1)C(=O)c1cccc(C#N)c1.CN(Cc1ccc(C(=O)N2CCCC3CCCCC32)cc1)C(=O)c1cccc(F)c1.CN(Cc1ccc(C(=O)N2CCCC3CCCCC32)cc1)C(=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HSD11B1 P28845 4/20 0.40
CNR2 P34972 1/20 0.40
HSD17B1 P14061 1/20 0.40
HTT P42858 1/20 0.39
CASR P41180 1/20 0.39
CYP3A4 P08684 5/20 0.38
USP2 O75604 4/20 0.38
CYP2D6 P10635 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
GLA P06280 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HPGD P15428 1/20 0.37
HCRTR1 O43613 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3811232 0.87 CNR2 (0.45) NSD2TDP1HSD11B1CNR2HSD17B1
SCHEMBL3811387 0.85 HSD11B1 (0.53) TDP1KDM4EHSD11B1CNR2HSD17B1
SCHEMBL3815228 0.83 NSD2 (0.47) NSD2CYP3A4ALDH1A1CYP2C19CYP2C9
SCHEMBL3810933 0.81 KMT2A (0.48) TDP1KDM4EHSD11B1HTTALDH1A1
SCHEMBL3810934 0.80 HSD11B1 (0.56) TDP1HSD11B1HSD17B1KMT2ASMN1; SMN2
SCHEMBL3818382 0.75 HDAC1 (0.55) ALDH1A1TSHRHPGDKMT2ALIMK2
SCHEMBL3813361 0.74 NSD2 (0.49) NSD2ALDH1A1HPGDKMT2A
SCHEMBL3814572 0.73 NSD2 (0.42) NSD2CNR2CASRMAPK1HCRTR1
SCHEMBL3813497 0.72 SMN1; SMN2 (0.55) TDP1HTTALDH1A1HPGDKMT2A
SCHEMBL3809571 0.70 KMT2A (0.42) HTTUSP2ALDH1A1MAPK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948190-A2 PHARMACEUTICAL USE OF SUBSTITUTED AMIDES TRANSTECH PHARMA (US) 2008-07-30 EP disclosed
WO-2007051810-A2 PHARMACEUTICAL USE OF SUBSTITUTED AMIDES TRANSTECH PHARMA (US) 2007-05-10 WO disclosed