SCHEMBL4608643

SCHEMBL4608643

NCc1ccc(C(F)(F)F)cc1-c1ccc(Br)cn1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.41
MPL P40238 2/20 0.36
MAOB P27338 1/20 0.36
FEN1 P39748 9/20 0.35
ALOX5AP P20292 8/20 0.35
THRB P10828 1/20 0.34
IDO1 P14902 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
STAT3 P40763 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836500 0.78 MEN1 (0.41) IDO1CYP1A2
SCHEMBL3713639 0.77 FEN1 (0.53) KDM1AMPLMAOBFEN1ALOX5AP
SCHEMBL20322968 0.71 KDM1A (0.53) KDM1AMAOBIDO1TRPV1
SCHEMBL31706466 0.70 IDO1 (0.43) MAOBIDO1
SCHEMBL18586785 0.68 KDM1A (0.45) KDM1AMPLFEN1ALOX5APCYP1A2
SCHEMBL12708057 0.67 IDO1 (0.43) MAOBIDO1
SCHEMBL29037326 0.66 IDO1 (0.37) MPLMAOBIDO1
SCHEMBL5466506 0.66 TRPV1 (0.41) MAOBIDO1TRPV1CYP1A2
Hydrochloric Acid SCHEMBL15021921 0.66 KCNA5 (0.43) MPLMAOBFEN1ALOX5APIDO1
SCHEMBL18587146 0.65 KDM1A (0.51) KDM1AMPLMAOBFEN1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885723-A2 PYRROLO[2,3-B]PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2008-02-13 EP disclosed
WO-2007013896-A2 PYRROL (2,3-B) PYRIDINE DERIVATIVES PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2007-02-01 WO disclosed