SCHEMBL460945

SCHEMBL460945

CN(C(=O)N1CCC(Nc2ccc(F)cc2)CC1)c1ccc(CN2CCN(C(=O)O)C(C(C)(C)C)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MLNR O43193 17/20 0.50
CYP3A4 P08684 7/20 0.50
CYP2D6 P10635 2/20 0.42
GHSR Q92847 1/20 0.42
KCNH2 Q12809 1/20 0.40
FAAH O00519 1/20 0.40
CCR5 P51681 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL377495 0.89 MLNR (0.54) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL460944 0.81 ALDH1A1 (0.55) MLNRCYP3A4
SCHEMBL377711 0.81 MLNR (0.74) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL378028 0.81 MLNR (0.60) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4210797 0.80 MLNR (0.55) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL378267 0.80 MLNR (0.55) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL1312338 0.79 MLNR (0.47) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1313152 0.78 MLNR (0.56) MLNRCYP3A4FAAHCCR5
SCHEMBL377818 0.78 MLNR (0.46) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL15152914 0.77 MLNR (0.56) MLNRCYP3A4CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029538-B1 BENZYLPIPERAZINE DERIVATIVES AS MOTILIN RECEPTOR ANTAGONISTS GLAXO GROUP LTD (GB) 2012-01-25 EP disclosed