SCHEMBL460958

SCHEMBL460958

COC(=O)N(Cc1cccc(F)c1)c1c(N)nc(-c2nn(Cc3ccccc3F)c3ncccc23)nc1N

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.73
KCNH2 Q12809 1/20 0.73
GUCY1A1 Q02108 12/20 0.52
GUCY1B1 Q02153 12/20 0.52
PDE5A O76074 6/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10062588 0.92 ADORA3 (0.76) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL459383 0.91 KCNH2 (0.81) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL10242938 0.88 ADORA3 (0.81) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL174905 0.86 KCNH2 (0.79) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL175338 0.86 ADORA3 (0.78) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL255819 0.86 ADORA3 (0.78) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
SCHEMBL256202 0.84 KCNH2 (0.84) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
Riociguat SCHEMBL245457 0.84 KCNH2 (1.00) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
Riociguat SCHEMBL29419573 0.84 KCNH2 (1.00) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A
Riociguat SCHEMBL29357210 0.84 KCNH2 (1.00) ADORA3KCNH2GUCY1A1GUCY1B1PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012010578-A1 SUBSTITUTED METHYL-PYRIMIDIN-5-YL CARBAMATES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-26 WO disclosed
WO-2012010578-A1 SUBSTITUTED METHYL-PYRIMIDIN-5-YL CARBAMATES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-26 WO disclosed