SCHEMBL4609592

SCHEMBL4609592

Cc1ccccc1C(OC[C@H]1CO1)C1CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
GLA P06280 1/20 0.47
KDM4E B2RXH2 1/20 0.46
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
CASR P41180 5/20 0.41
CYP2D6 P10635 3/20 0.41
TDP1 Q9NUW8 1/20 0.40
ESR1 P03372 1/20 0.37
TP53 P04637 3/20 0.36
TSHR P16473 3/20 0.36
CYP3A4 P08684 2/20 0.36
HIF1A Q16665 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
IDO1 P14902 1/20 0.33
CHRNA7 P36544 1/20 0.33
SLC22A2 O15244 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14502702 1.00 ALDH1A1 (0.47) ALDH1A1GLAKDM4ESLC6A2SLC6A4
SCHEMBL4609594 1.00 ALDH1A1 (0.47) ALDH1A1GLAKDM4ESLC6A2SLC6A4
SCHEMBL29267774 0.86 ALDH1A1 (0.49) ALDH1A1GLAKDM4ESLC6A2SLC6A4
SCHEMBL4610221 0.85 ALDH1A1 (0.45) ALDH1A1GLAKDM4ESLC6A2SLC6A4
SCHEMBL14502704 0.85 ALDH1A1 (0.45) ALDH1A1GLAKDM4ESLC6A2SLC6A4
SCHEMBL4610224 0.85 ALDH1A1 (0.45) ALDH1A1GLAKDM4ESLC6A2SLC6A4
SCHEMBL17226943 0.84 TDP1 (0.39) ALDH1A1GLAKDM4ETDP1TP53
SCHEMBL6742323 0.84 TDP1 (0.39) ALDH1A1GLAKDM4ETDP1TP53
SCHEMBL6743415 0.84 TDP1 (0.39) ALDH1A1GLAKDM4ETDP1TP53
SCHEMBL4610991 0.80 ALDH1A1 (0.51) ALDH1A1GLASLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1308436-B1 CALCIUM RECEPTOR ANTAGONISTS JAPAN TOBACCO INC (JP) 2008-10-15 EP disclosed
US-7211685-B2 Calcium receptor antagonists JAPAN TOBACCO INC. (JP) 2007-05-01 US disclosed
US-7211685-B2 Calcium receptor antagonists JAPAN TOBACCO INC. (JP) 2007-05-01 US disclosed
US-7211685-B2 Calcium receptor antagonists JAPAN TOBACCO INC. (JP) 2007-05-01 US disclosed
US-6916956-B2 Calcium receptor antagonist JAPAN TOBACCO, INC. (JP) 2005-07-12 US disclosed
US-20050107448-A1 Calcium receptor antagonists JAPAN TABACCO INC. 2005-05-19 US disclosed
US-20040006130-A1 Calcium receptor antagonist JAPAN TOBACCO INC (JP) 2004-01-08 US disclosed
EP-1308436-A1 CALCIUM RECEPTOR ANTAGONISTS JAPAN TOBACCO INC. (JP) 2003-05-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050107448-A1 Calcium receptor antagonists CASR, CALCR, CALCRL ALDH1A1 4104/4885GLA 2441/4885KDM4E 2372/4885
US-20040006130-A1 Calcium receptor antagonist CALCRL, CASR, CALCR ALDH1A1 3406/4885GLA 2049/4885KDM4E 2199/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.