SCHEMBL4609643

SCHEMBL4609643

Nc1cc(O)nc(O)c1N

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30964214 0.79 MAPT (0.32) KDM4EALDH1A1LMNAGAAMAPT
SCHEMBL3367926 0.79 NQO1 (0.33) KDM4EALDH1A1LMNAGAAMAPT
SCHEMBL5705216 0.79 MAPT (0.32) KDM4EALDH1A1LMNAGAAMAPT
SCHEMBL2905943 0.75
SCHEMBL11777661 0.70 POLB (0.36) LMNA
Sulfuric Acid SCHEMBL2398134 0.69 NT5E (0.34) KDM4EALDH1A1GAAMAPT
SCHEMBL7690577 0.65
SCHEMBL29140679 0.65 PTK2 (0.44) KDM4EALDH1A1LMNAGAAMAPT
SCHEMBL9794284 0.65
SCHEMBL8517257 0.63 MAPT (0.32) ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 195 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1231889-B1 DIRECT HAIR DYES AND USE THEREOF HENKEL KGAA (DE) 2005-12-14 EP claimed
EP-1309540-B1 OXIDIZING COLORANT HENKEL KGAA (DE) 2005-11-02 EP claimed
EP-0988022-B1 HAIR DYE HENKEL KGAA (DE) 2005-09-21 EP claimed
EP-1212032-B1 NEW DIRECT HAIR COLORANTS HENKEL KGAA (DE) 2005-05-04 EP claimed
US-20040261198-A1 Restructuring and finishing of keratin fibers HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (HENKEL KGAA) (DE) 2004-12-30 US claimed
US-6835211-B1 Comprises 1,4-dihydroxy-6-chloro-7-(3'-methylphenoxy)-anthraquinone; improved colorfastness HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2004-12-28 US claimed
US-6818023-B2 CONTAINING AN INDOLINE, AN INDOLE, OR A DERIVATIVE THEREOF IN COMBINATION WITH AT LEAST ONE AMINO ACID OR OLIGOPEPTIDE. HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2004-11-16 US claimed
US-6814761-B1 Direct hair colorants HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2004-11-09 US claimed
EP-1210060-B1 DEVELOPER-COUPLER COMBINATIONS HENKEL KGAA (DE) 2004-09-15 EP claimed
EP-1455736-A1 RESTRUCTURING AND FINISHING OF KERATIN FIBERS Henkel Kommanditgesellschaft auf Aktien (DE) 2004-09-15 EP claimed
WO-2001000142-A2 DEVELOPER-COUPLER COMBINATIONS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2001-01-04 WO claimed
WO-2000061090-A1 METHOD AND COLORANT FOR DYEING KERATIN FIBERS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2000-10-19 WO claimed
WO-2000061088-A1 COLORANTS CONTAINING 4-AMINO-2-AMINOMETHYL-PHENOL DERIVATIVES AND THEIR USE FOR COLORING KERATIN FIBERS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2000-10-19 WO claimed
WO-2000021497-A1 COLOURING AGENTS WITH ENZYMES HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2000-04-20 WO claimed
EP-0988022-A1 HAIR DYE Henkel Kommanditgesellschaft auf Aktien (DE) 2000-03-29 EP claimed
WO-1999066890-A1 COLORANT FOR COLOURING KERATIN FIBRES HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1999-12-29 WO claimed
WO-1999066889-A1 NEW COUPLING COMPONENTS FOR OXIDATION HAIR COLOURING PRODUCTS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1999-12-29 WO claimed
WO-1999065891-A1 NOVEL 2,4-DIAMINOPHENOL DERIVATIVES AND THE USE THEREOF HANS SCHWARZKOPF GMBH & CO. KG (DE) 1999-12-23 WO claimed
WO-1999065865-A1 NOVEL 3,4-DIAMINOPHENOL DERIVATIVES AND THEIR USE HANS SCHWARZKOPF GMBH & CO. KG (DE) 1999-12-23 WO claimed
WO-1999007334-A1 HAIR DYE HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1999-02-18 WO claimed