SCHEMBL461324

SCHEMBL461324

Cc1nn(-c2ccc(C#N)c(NC3CCC(O)CC3)c2)c2cccc(-c3nc4ccc(F)cc4[nH]3)c12

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 15/20 0.49
HSP90AB1 P08238 8/20 0.35
AMY1A P0DUB6 2/20 0.35
PDE10A Q9Y233 1/20 0.34
PRKCQ Q04759 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL461325 1.00 HSP90AA1 (0.49) HSP90AA1HSP90AB1AMY1APDE10APRKCQ
SCHEMBL461822 0.90 HSP90AA1 (0.42) HSP90AA1HSP90AB1AMY1APRKCQ
SCHEMBL461821 0.90 HSP90AA1 (0.42) HSP90AA1HSP90AB1AMY1APRKCQ
SCHEMBL1076054 0.87 HSP90AA1 (0.36) HSP90AA1HSP90AB1AMY1APRKCQ
SCHEMBL463010 0.86 HSP90AA1 (0.66) HSP90AA1HSP90AB1
SCHEMBL463009 0.86 HSP90AA1 (0.66) HSP90AA1HSP90AB1
SCHEMBL2181661 0.85 HSP90AA1 (0.36) HSP90AA1AMY1APRKCQ
SCHEMBL1076728 0.85 AMY1A (0.35) HSP90AA1AMY1APDE10APRKCQ
SCHEMBL383558 0.83 AR (0.36) HSP90AA1AMY1APDE10A
SCHEMBL1078057 0.83 HSP90AA1 (0.47) HSP90AA1AMY1APRKCQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408762-A1 HSP90 INHIBITING INDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING SAME AND USE THEREOF SANOFI (FR) 2012-01-25 EP disclosed
WO-2010106290-A1 HSP90 INHIBITING INDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING SAME AND USE THEREOF SANOFI-AVENTIS (FR) 2010-09-23 WO disclosed