SCHEMBL4613677

SCHEMBL4613677

O=c1[nH]c(=O)n(CC2CC2)c2nc(C(Cc3ccccc3F)c3ccc(NS(=O)(=O)c4cnc(Cl)c(Br)c4)cc3)[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PCK1 P35558 13/20 0.42
HTT P42858 1/20 0.34
ALDH1A1 P00352 3/20 0.33
EIF2AK3 Q9NZJ5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4612950 0.86 PCK1 (0.45) PCK1
SCHEMBL4612921 0.85 PCK1 (0.58) PCK1
SCHEMBL4614243 0.83 PCK1 (0.53) PCK1
SCHEMBL4614318 0.83 PCK1 (0.43) PCK1ALDH1A1
SCHEMBL4613199 0.83 PCK1 (0.47) PCK1ALDH1A1
SCHEMBL4612956 0.82 PCK1 (0.55) PCK1
SCHEMBL4614233 0.82 PCK1 (0.47) PCK1ALDH1A1
SCHEMBL4615362 0.81 PCK1 (0.60) PCK1
SCHEMBL4614242 0.81 PCK1 (0.58) PCK1
SCHEMBL6279236 0.81 PCK1 (0.42) PCK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599477-B1 SULFONAMIDE SUBSTITUTED XANTHINE DERIVATIVES FOR USE AS PEPCK INHIBITORS HOFFMANN LA ROCHE (CH) 2008-01-30 EP claimed