SCHEMBL46164

SCHEMBL46164

O=C(c1nc(-c2cccc(-c3cn4ncccc4n3)c2)no1)N1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.43
SMN1; SMN2 Q16637 6/20 0.41
PDE4B Q07343 4/20 0.40
PDE4D Q08499 3/20 0.40
KCNH2 Q12809 1/20 0.40
MCHR1 Q99705 1/20 0.40
NPC1 O15118 8/20 0.39
RAB9A P51151 7/20 0.39
HPGD P15428 6/20 0.39
ALDH1A1 P00352 4/20 0.39
TP53 P04637 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPK1 P28482 2/20 0.39
TSHR P16473 2/20 0.39
NFKB1 P19838 2/20 0.39
NFKB2 Q00653 2/20 0.39
RELA Q04206 2/20 0.39
PDE4A P27815 2/20 0.39
PDE4C Q08493 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL45311 0.99 SMN1; SMN2 (0.41) GRM5SMN1; SMN2PDE4BPDE4DKCNH2
SCHEMBL45748 0.91 CYP1A2 (0.43) SMN1; SMN2NPC1RAB9AHPGDALDH1A1
SCHEMBL44385 0.88 KMT2A (0.40) SMN1; SMN2KCNH2MCHR1NPC1RAB9A
SCHEMBL44578 0.84 RAB9A (0.40) SMN1; SMN2NPC1RAB9A
SCHEMBL44170 0.83 GAA (0.41) SMN1; SMN2NPC1RAB9ATP53THRB
SCHEMBL44476 0.81 GAA (0.37) SMN1; SMN2NPC1RAB9AHPGDALDH1A1
SCHEMBL43913 0.81 GAA (0.43) SMN1; SMN2NPC1RAB9AHPGDALDH1A1
SCHEMBL44367 0.80 NPC1 (0.43) SMN1; SMN2PDE4BPDE4DNPC1RAB9A
SCHEMBL44764 0.78 GAA (0.44) TP53KMT2ATHRB
SCHEMBL43972 0.78 HTT (0.53) SMN1; SMN2KCNH2TP53MAPK1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed