SCHEMBL4619911

SCHEMBL4619911

O=[N+]([O-])/C=C/c1cccc(OCF)c1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 12/20 0.70
TLR2 O60603 12/20 0.70
MAOA P21397 9/20 0.68
MAOB P27338 9/20 0.68
FBP1 P09467 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4619916 1.00 TLR4 (0.70) TLR4TLR2MAOAMAOBFBP1
SCHEMBL2539612 0.84 MAOA (0.70) TLR4TLR2MAOAMAOBFBP1
SCHEMBL1967344 0.83 TLR4 (0.67) TLR4TLR2MAOAMAOBFBP1
SCHEMBL1967341 0.83 TLR4 (0.67) TLR4TLR2MAOAMAOBFBP1
SCHEMBL510207 0.82 TLR4 (1.00) TLR4TLR2MAOAMAOBFBP1
SCHEMBL510208 0.82 TLR4 (1.00) TLR4TLR2MAOAMAOBFBP1
SCHEMBL510222 0.81 MAOA (1.00) TLR4TLR2MAOAMAOB
SCHEMBL510223 0.81 MAOA (1.00) TLR4TLR2MAOAMAOB
SCHEMBL18177331 0.81 TLR4 (0.67) TLR4TLR2MAOAMAOBFBP1
SCHEMBL510378 0.80 TLR4 (1.00) TLR4TLR2MAOAMAOBFBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019200120-A1 DIHYDROISOQUINOLINE-2(1H)-CARBOXAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS LYCERA CORPORATION (US) 2019-10-17 WO disclosed
WO-2008039882-A1 A COMBINATION OF NIACIN AND A PROSTAGLANDIN D2 RECEPTOR ANTAGONIST SANOFI-AVENTIS U.S. LLC (US) 2008-04-03 WO disclosed
EP-1891019-A2 2,6-SUBSTITUTED-4-MONOSUBSTITUTEDAMINO-PYRIMIDINE AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS Aventis Pharmaceuticals Inc. (US) 2008-02-27 EP disclosed
WO-2006044732-A2 2, 6-SUBSTITUTED-4-MONOSUBSTITUTEDAMINO-PYRIMIDINE AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2006-04-27 WO disclosed