SCHEMBL4621653

SCHEMBL4621653

CCOc1cccc(S(=O)(=O)N2CCC(N3C(=O)OCc4cccc(C)c43)CC2)c1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 9/20 0.63
OXTR P30559 1/20 0.44
KDM4E B2RXH2 2/20 0.41
TSHR P16473 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3137315 0.90 HTR6 (0.77) HTR6OXTRTSHRALDH1A1
SCHEMBL3152345 0.86 HTR6 (0.68) HTR6
SCHEMBL3148210 0.85 HTR6 (0.74) HTR6ALDH1A1
SCHEMBL3146923 0.84 HTR6 (0.66) HTR6ALDH1A1
SCHEMBL3138605 0.84 HTR6 (0.66) HTR6SMN1; SMN2
SCHEMBL3148297 0.84 HTR6 (0.66) HTR6KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3142878 0.84 HTR6 (0.68) HTR6ALDH1A1
SCHEMBL3152438 0.83 HTR6 (0.73) HTR6KDM4EALDH1A1SMN1; SMN2
SCHEMBL3152654 0.83 HTR6 (0.66) HTR6ALDH1A1SMN1; SMN2
SCHEMBL3148124 0.82 HTR6 (0.66) HTR6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902733-A1 Combination of a NMDA-receptor ligand and a compound with 5-HT6 receptor affinity LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2008-03-26 EP disclosed