SCHEMBL462374

SCHEMBL462374

COc1cccc(C(=O)NC2CNc3ccc(C(=O)O)cc3C2)c1

nearest known ligand 0.86

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 10/20 0.86
GRM5 P41594 1/20 0.48
ALDH1A1 P00352 2/20 0.47
TSHR P16473 1/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 1/20 0.46
MAPK1 P28482 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM5A P29375 1/20 0.45
MCHR1 Q99705 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10192710 0.93 HDAC8 (0.85) HDAC8GRM5ALDH1A1TSHRNPC1
SCHEMBL443998 0.93 HDAC8 (1.00) HDAC8GRM5ALDH1A1TSHRMEN1
SCHEMBL461269 0.79 HDAC8 (0.85) HDAC8TSHRMAPK1MEN1KMT2A
SCHEMBL445401 0.76 HDAC8 (1.00) HDAC8GRM5NPC1RAB9AMEN1
SCHEMBL443999 0.76 HDAC8 (0.52) HDAC8GRM5ALDH1A1TSHRNPC1
SCHEMBL2468483 0.75 NPC1 (0.71) GRM5ALDH1A1TSHRNPC1RAB9A
SCHEMBL444288 0.75 HDAC8 (1.00) HDAC8NPC1RAB9AMEN1KMT2A
SCHEMBL444916 0.74 HDAC8 (1.00) HDAC8ALDH1A1MEN1KMT2A
SCHEMBL3619472 0.73 HDAC8 (0.49) HDAC8NPC1RAB9AMEN1KMT2A
SCHEMBL10247271 0.73 HDAC8 (0.68) HDAC8GRM5ALDH1A1TSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2613775-A1 NOVEL N-HYDROXY-BENZAMIDES FOR THE TREATMENT OF CANCER F.HOFFMANN-LA ROCHE AG (CH) 2013-07-17 EP claimed
WO-2012031993-A1 NOVEL N-HYDROXY-BENZAMIDES FOR THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2012-03-15 WO claimed