SCHEMBL4623907

SCHEMBL4623907

CCOC(=O)C(C#N)=C(O)C(F)(F)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
TSHR P16473 1/20 0.44
CES2 O00748 5/20 0.44
CES1 P23141 5/20 0.44
CYP2C9 P11712 1/20 0.39
MAPT P10636 5/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.35
ACHE P22303 4/20 0.35
USP2 O75604 1/20 0.33
LMNA P02545 1/20 0.33
CRHBP P24387 1/20 0.33
RAB9A P51151 1/20 0.33
CRHR2 Q13324 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4623904 1.00 ALDH1A1 (0.44) ALDH1A1TSHRCES2CES1CYP2C9
SCHEMBL7853979 0.86 ALDH1A1 (0.47) ALDH1A1TSHRCES2CES1CYP2C9
SCHEMBL7853980 0.86 ALDH1A1 (0.47) ALDH1A1TSHRCES2CES1CYP2C9
SCHEMBL2592394 0.85 ALDH1A1 (0.46) ALDH1A1TSHRCES2CES1CYP2C9
SCHEMBL2592388 0.85 ALDH1A1 (0.46) ALDH1A1TSHRCES2CES1CYP2C9
SCHEMBL13237290 0.81 ALDH1A1 (0.48) ALDH1A1TSHRCYP2C9MAPTMEN1
SCHEMBL1754710 0.78 ALDH1A1 (0.61) ALDH1A1TSHRCYP2C9MAPTMEN1
SCHEMBL2115865 0.78 ALDH1A1 (0.61) ALDH1A1TSHRCYP2C9MAPTMEN1
SCHEMBL20551568 0.76 ALDH1A1 (0.47) ALDH1A1TSHRCYP2C9MAPTMEN1
SCHEMBL4625344 0.75 ALDH1A1 (0.46) ALDH1A1TSHRCYP2C9MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1067121-B1 5-Aminopyrazole-4-carboxylate derivative and process for preparing the same MITSUI CHEMICALS INC (JP) 2008-05-28 EP disclosed
US-6235911-B1 5-aminopyrazole-4-carboxylate derivative and process for preparing the same MITSUI CHEMICALS, INC. (JP) 2001-05-22 US disclosed
EP-1067121-A2 5-Aminopyrazole-4-carboxylate derivative and process for preparing the same Mitsui Chemicals, Inc. (JP) 2001-01-10 EP disclosed