SCHEMBL4625161

SCHEMBL4625161

CC(c1ccc2nc(-c3c(Cl)cccc3Cl)ccc2c1)C(NC(=O)c1ccc(N)nc1)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.45
ITGAV P06756 1/20 0.45
HPGDS O60760 5/20 0.40
ABL1 P00519 3/20 0.39
GPR132 Q9UNW8 1/20 0.36
EPHX2 P34913 2/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CCKAR P32238 2/20 0.34
CCKBR P32239 2/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MAP4K4 O95819 1/20 0.34
DGAT1 O75907 1/20 0.34
BCR P11274 2/20 0.33
S1PR2 O95136 1/20 0.33
S1PR4 O95977 1/20 0.33
S1PR3 Q99500 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3319927 0.84 ITGB1 (0.62) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL1028110 0.83 ITGB1 (0.55) ITGB1ITGAVABL1GPR132CCKAR
SCHEMBL4625016 0.80 ITGB1 (0.72) ITGB1ITGAVHPGDSCA1CA2
SCHEMBL3313211 0.79 ITGB1 (0.51) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL3314603 0.78 ITGB1 (0.45) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL1030227 0.78 ITGB1 (0.46) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL6151284 0.77 ITGB1 (0.47) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL4625157 0.76 ITGB1 (0.59) ITGB1ITGAVHPGDSABL1EPHX2
SCHEMBL4624866 0.76 ITGB1 (0.52) ITGB1ITGAVCCKARCCKBR
SCHEMBL4750012 0.76 ITGB1 (0.49) ITGB1ITGAVABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP disclosed