SCHEMBL6151284

SCHEMBL6151284

CC(c1ccc2nc(-c3c(Cl)cccc3Cl)ccc2c1)C(NC(=O)C1(N)CCCC1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.47
ITGAV P06756 1/20 0.47
ABL1 P00519 1/20 0.40
AKT1 P31749 7/20 0.33
RPS6KB1 P23443 3/20 0.33
CCKAR P32238 2/20 0.32
CCKBR P32239 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
ROCK2 O75116 5/20 0.32
AKT2 P31751 5/20 0.32
AKT3 Q9Y243 5/20 0.32
KCNH2 Q12809 4/20 0.32
PRCP P42785 2/20 0.31
ITGA4 P13612 2/20 0.31
ITGB7 P26010 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5173387 0.86 ITGB1 (0.44) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL3319927 0.82 ITGB1 (0.62) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL3320918 0.80 ITGB1 (0.70) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL1028110 0.79 ITGB1 (0.55) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL1030227 0.79 ITGB1 (0.46) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL3315803 0.79 ALDH1A1 (0.37) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL4750012 0.77 ITGB1 (0.49) ITGB1ITGAVABL1CYP1A2CYP2C9
SCHEMBL4626500 0.77 ITGB1 (0.49) ITGB1ITGAVABL1CYP1A2CYP2C9
SCHEMBL4625161 0.77 ITGB1 (0.45) ITGB1ITGAVABL1CCKARCCKBR
SCHEMBL3313211 0.77 ITGB1 (0.51) ITGB1ITGAVABL1CCKARCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed