SCHEMBL4625253

SCHEMBL4625253

Cc1ccc(S(=O)(=O)N2C(C(=O)NC(Cc3ccc4nc(-c5cc(C(F)(F)F)ccc5Cl)ccc4c3)C(=O)O)CC3CCCC[C@@H]32)cc1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 13/20 0.43
ITGA4 P13612 13/20 0.43
ALDH1A1 P00352 1/20 0.40
ITGAV P06756 1/20 0.37
TRPA1 O75762 2/20 0.36
ITGB7 P26010 1/20 0.36
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3313128 1.00 ITGB1 (0.43) ITGB1ITGA4ALDH1A1ITGAVTRPA1
SCHEMBL3314360 0.90 ITGB1 (0.48) ITGB1ITGA4ALDH1A1ITGAVITGB7
SCHEMBL3313932 0.89 ITGA4 (0.46) ITGB1ITGA4ALDH1A1ITGAVITGB7
SCHEMBL4410500 0.86 ITGB1 (0.53) ITGB1ITGA4ALDH1A1ITGAVITGB7
SCHEMBL3317863 0.86 ITGB1 (0.53) ITGB1ITGA4ALDH1A1ITGAVITGB7
SCHEMBL3318694 0.85 ITGB1 (0.45) ITGB1ITGA4ALDH1A1ITGAVITGB7
SCHEMBL6141601 0.81 ITGB1 (0.39) ITGB1ITGA4ALDH1A1ITGAV
SCHEMBL4625418 0.80 ITGB1 (0.44) ITGB1ITGA4ALDH1A1ITGAVITGB7
SCHEMBL3320849 0.74 ITGB1 (0.56) ITGB1ITGA4ALDH1A1ITGAVITGB7
SCHEMBL3314257 0.74 ITGB1 (0.51) ITGB1ITGA4ITGAVITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP disclosed