SCHEMBL4627713

SCHEMBL4627713

O=S(=O)(c1ccc(-c2ccccn2)s1)N1CCNCC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
GHSR Q92847 4/20 0.55
POLB P06746 1/20 0.53
KMT2A Q03164 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
MMP8 P22894 2/20 0.47
MMP3 P08254 2/20 0.47
PKM P14618 1/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
NPC1 O15118 1/20 0.46
GLA P06280 1/20 0.46
RAB9A P51151 1/20 0.46
MMP1 P03956 1/20 0.45
MMP2 P08253 1/20 0.45
MMP7 P09237 1/20 0.45
CYP3A4 P08684 1/20 0.45
TSHR P16473 1/20 0.45
NFKB1 P19838 1/20 0.45
THPO P40225 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15958829 0.80 ALDH1A1 (0.64) ALDH1A1GHSRPOLBKMT2AL3MBTL1
Hydrochloric Acid SCHEMBL1314648 0.79 ALDH1A1 (0.63) ALDH1A1GHSRPOLBKMT2AL3MBTL1
SCHEMBL6184020 0.76 IKBKB (0.61) PKMMAPT
SCHEMBL1314374 0.75 ALDH1A1 (0.63) ALDH1A1GHSRPOLBKMT2AL3MBTL1
SCHEMBL1314372 0.75 ALDH1A1 (0.66) ALDH1A1POLBKMT2AL3MBTL1MMP8
SCHEMBL14055914 0.73 ALDH1A1 (0.59) ALDH1A1POLBKMT2AL3MBTL1MMP8
SCHEMBL1618671 0.73 ALDH1A1 (0.52) ALDH1A1POLBKMT2AL3MBTL1MMP8
SCHEMBL15462054 0.73 ALDH1A1 (0.53) ALDH1A1GHSRPOLBKMT2AL3MBTL1
SCHEMBL1619096 0.73 HDAC1 (0.56) ALDH1A1POLBKMT2AL3MBTL1MMP8
SCHEMBL3055723 0.72 KDM4E (0.60) ALDH1A1POLBL3MBTL1MMP8MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981848-A2 11-BETA HSD1 INHIBITORS Wyeth (US) 2008-10-22 EP disclosed
WO-2007092435-A2 11-BETA HSD1 INHIBITORS WYETH (US) 2007-08-16 WO disclosed