SCHEMBL4627715

SCHEMBL4627715

CC(C)(C)OC(=O)NC(Cc1ccc2nc(-c3ccccc3)ccc2c1)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.58
CTSS P25774 5/20 0.56
CTSK P43235 4/20 0.56
CTSB P07858 3/20 0.56
ACE P12821 1/20 0.55
ITGB1 P05556 2/20 0.52
ITGAV P06756 2/20 0.52
PIN1 Q13526 2/20 0.48
PPARA Q07869 5/20 0.48
PPARG P37231 4/20 0.48
ITGB3 P05106 2/20 0.48
ITGA2B P08514 2/20 0.48
PPARD Q03181 2/20 0.47
CTSL P07711 1/20 0.47
ITGA4 P13612 1/20 0.46
ITGB7 P26010 1/20 0.46
ITGB5 P18084 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3316089 0.92 CTSS (0.54) PTPN1CTSSCTSKCTSBACE
SCHEMBL3317745 0.88 ITGB1 (0.56) PTPN1CTSSCTSKCTSBACE
SCHEMBL3315439 0.87 ITGB1 (0.71) PTPN1CTSSCTSKCTSBACE
SCHEMBL3318595 0.87 ITGB1 (0.71) PTPN1CTSSCTSKCTSBACE
SCHEMBL4626858 0.87 ITGB1 (0.71) PTPN1CTSSCTSKCTSBACE
SCHEMBL4627669 0.86 ITGB1 (0.55) PTPN1CTSSCTSKCTSBACE
SCHEMBL3315927 0.86 ITGB1 (0.55) PTPN1CTSSCTSKCTSBACE
SCHEMBL3314031 0.86 ITGB1 (0.55) PTPN1CTSSCTSKCTSBACE
SCHEMBL4627618 0.85 PTPN1 (0.58) PTPN1CTSSCTSKCTSBACE
SCHEMBL3318761 0.84 ITGB1 (0.59) PTPN1CTSSCTSKCTSBACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP claimed