SCHEMBL4628756

SCHEMBL4628756

COc1ccc(C(=O)NC(=N)Nc2cc(OC)c(OC)c(OC)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.56
SMN1; SMN2 Q16637 4/20 0.56
NPC1 O15118 3/20 0.56
RAB9A P51151 3/20 0.56
ALDH1A1 P00352 3/20 0.56
ATM Q13315 1/20 0.55
GAA P10253 4/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
TUBB4A P04350 1/20 0.54
TUBB P07437 1/20 0.54
TUBA3C P0DPH7 1/20 0.54
TUBA1B P68363 1/20 0.54
TUBA4A P68366 1/20 0.54
TUBB4B P68371 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4628461 0.90 SCN5A (0.57) TP53SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL4628473 0.89 MAPT (0.56) TP53SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL8224616 0.87 SMO (0.65) TP53SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL5276408 0.87 SMN1; SMN2 (0.48) SMN1; SMN2RAB9AATMGAAMEN1
SCHEMBL9190300 0.86 TP53 (0.73) TP53SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL4628525 0.81 TUBB4A (0.51) SMN1; SMN2NPC1RAB9AALDH1A1MEN1
SCHEMBL11911362 0.81 SMO (0.60) ALDH1A1MEN1KMT2ACYP3A4CYP1A2
SCHEMBL4627489 0.79 ABCB1 (0.55) TP53SMN1; SMN2ALDH1A1GAAMEN1
SCHEMBL8224334 0.79 SMO (0.66) SMN1; SMN2ALDH1A1GAAMEN1KMT2A
SCHEMBL4104318 0.77 SMN1; SMN2 (0.51) TP53SMN1; SMN2ALDH1A1ATMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032556-B1 PHARMACEUTICALLY ACTIVE COMPOUNDS AND METHODS OF USE WYETH CORP (US) 2007-12-19 EP claimed
US-7041702-B1 Pharmaceutically active compounds and methods of use SCION PHARMACEUTICALS, INC. (US) 2006-05-09 US claimed
EP-1918272-A1 Pharmaceutically active compounds and methods of use Wyeth a Corporation of the State of Delaware (US) 2008-05-07 EP disclosed
EP-1032556-B1 PHARMACEUTICALLY ACTIVE COMPOUNDS AND METHODS OF USE WYETH CORP (US) 2007-12-19 EP disclosed
US-20060270741-A1 Pharmaceutically active compounds and methods of use SCION PHARMACEUTICALS, INC. (US) 2006-11-30 US disclosed
US-7041702-B1 Pharmaceutically active compounds and methods of use SCION PHARMACEUTICALS, INC. (US) 2006-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060270741-A1 Pharmaceutically active compounds and methods of use GBA1, CTSA, GAA TP53 4226/4885SMN1; SMN2 53/4885NPC1 140/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.