SCHEMBL4629679

SCHEMBL4629679

Clc1ccc(CC2=NCCN2)cc1Cl.Clc1cccc(Cl)c1CC1=NCCN1

nearest known ligand 0.76

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 8/20 0.76
HTR1B P28222 5/20 0.55
CYP2D6 P10635 3/20 0.55
NFKB1 P19838 1/20 0.55
HTR1D P28221 7/20 0.51
CYP1A2 P05177 2/20 0.51
ADRA2A P08913 2/20 0.51
ADRA2B P18089 2/20 0.51
ADRA2C P18825 2/20 0.51
ADRA1D P25100 2/20 0.51
ADRA1A P35348 2/20 0.51
ADRA1B P35368 2/20 0.51
LMNA P02545 1/20 0.51
TSHR P16473 1/20 0.51
HIF1A Q16665 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL953553 0.90 TAAR1 (0.60) TAAR1HTR1BCYP2D6NFKB1HTR1D
SCHEMBL955616 0.87 TAAR1 (1.00) TAAR1HTR1BCYP2D6NFKB1HTR1D
SCHEMBL4630000 0.79 TAAR1 (0.82) TAAR1HTR1BCYP2D6NFKB1HTR1D
SCHEMBL21519443 0.78 TAAR1 (0.81) TAAR1HTR1BCYP2D6HTR1DCYP1A2
SCHEMBL956643 0.77 TAAR1 (0.79) TAAR1HTR1BCYP2D6HTR1DCYP1A2
SCHEMBL952955 0.77 TAAR1 (0.79) TAAR1HTR1BCYP2D6NFKB1HTR1D
SCHEMBL26078508 0.77 TAAR1 (0.79) TAAR1HTR1BCYP2D6NFKB1HTR1D
SCHEMBL4986025 0.77 TAAR1 (0.56) TAAR1HTR1BCYP2D6NFKB1HTR1D
Hydrochloric Acid SCHEMBL956502 0.76 TAAR1 (0.77) TAAR1HTR1BCYP2D6HTR1DCYP1A2
SCHEMBL953728 0.74 TAAR1 (0.73) TAAR1HTR1BCYP2D6NFKB1HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP claimed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO claimed
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed