SCHEMBL4629994

SCHEMBL4629994

COc1cccc(CCCCCN)c1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA14 Q9ULX7 1/20 0.52
TAAR1 Q96RJ0 1/20 0.51
CHRM2 P08172 1/20 0.50
ABCB1 P08183 3/20 0.48
ALOX5 P09917 1/20 0.47
PTGS2 P35354 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
PPARA Q07869 1/20 0.46
ACHE P22303 1/20 0.43
CYP1A2 P05177 1/20 0.42
GAA P10253 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
TSHR P16473 1/20 0.42
CRHBP P24387 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL558962 0.98 CA12 (0.54) CA12CA1CA2CA14TAAR1
SCHEMBL15610427 0.93 CA12 (0.55) CA12CA1CA2CA14TAAR1
SCHEMBL30839502 0.86 TAAR1 (0.69) CA12CA1CA2CA14TAAR1
SCHEMBL151944 0.86 TAAR1 (0.69) CA12CA1CA2CA14TAAR1
SCHEMBL9238920 0.85 ALOX5 (0.66) CA12CA1CA2CA14ABCB1
SCHEMBL15206587 0.85 ALOX5 (0.66) CA12CA1CA2CA14ABCB1
SCHEMBL15656477 0.85 ALOX5 (0.66) CA12CA1CA2CA14ABCB1
SCHEMBL28772139 0.85 ALOX5 (0.66) CA12CA1CA2CA14ABCB1
SCHEMBL9118416 0.85 ALOX5 (0.66) CA12CA1CA2CA14ABCB1
SCHEMBL15658926 0.85 ALOX5 (0.66) CA12CA1CA2CA14ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517883-B8 ORTHO-SUBSTITUTED BENZOIC ACID DERIVATIVES FOR THE TREATMENT OF INSULIN RESISTANCE ASTRAZENECA AB (SE) 2008-05-21 EP disclosed
EP-1517883-A1 ORTHO-SUBSTITUTED BENZOIC ACID DERIVATIVES FOR THE TREATMENT OF INSULIN RESISTANCE AstraZeneca AB (SE) 2005-03-30 EP disclosed
WO-2004000790-A1 ORTHO-SUBSTITUTED BENZOIC ACID DERIVATIVES FOR THE TREATMENT OF INSULIN RESISTANCE ASTRAZENECA AB (SE) 2003-12-31 WO disclosed