SCHEMBL4630237

SCHEMBL4630237

CCOc1cc(CC)c(Cc2ncc[nH]2)c(CC)c1.CCOc1ccc(CC)c(Cc2ncc[nH]2)c1CC

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 6/20 0.56
HTR1A P08908 1/20 0.56
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
NAMPT P43490 2/20 0.31
VCP P55072 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL953854 0.92 TAAR1 (0.62) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL953241 0.88 TAAR1 (0.63) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL4630512 0.83 TAAR1 (0.57) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL4630242 0.82 TAAR1 (0.54) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL953878 0.81 TAAR1 (0.62) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL954135 0.80 TAAR1 (0.60) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL954171 0.78 TAAR1 (0.58) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL953613 0.77 TAAR1 (0.63) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL955275 0.76 TAAR1 (0.66) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL954953 0.75 TAAR1 (0.60) TAAR1HTR1AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed