SCHEMBL4630242

SCHEMBL4630242

CCOc1ccc(CC)c(Cc2ncc[nH]2)c1CC.CCc1ccc(OCc2ccccc2)c(CC)c1Cc1ncc[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 7/20 0.54
HTR1A P08908 2/20 0.54
AOC3 Q16853 1/20 0.41
MAPK14 Q16539 1/20 0.40
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
MAPK1 P28482 2/20 0.38
NTSR1 P30989 2/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
LMNA P02545 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.36
ADRA2A P08913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL954171 0.97 TAAR1 (0.58) TAAR1HTR1AAOC3MAPK14MAPK1
SCHEMBL953854 0.89 TAAR1 (0.62) TAAR1HTR1AAOC3MAPTHPGD
SCHEMBL954135 0.82 TAAR1 (0.60) TAAR1HTR1AKDM4EALDH1A1GAA
SCHEMBL4630237 0.82 TAAR1 (0.56) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL953878 0.80 TAAR1 (0.62) TAAR1HTR1AADRA1DADRA1AADRA1B
SCHEMBL954953 0.78 TAAR1 (0.60) TAAR1HTR1AL3MBTL1LMNAADRA2A
SCHEMBL9414540 0.74 TAAR1 (0.61) TAAR1HTR1AMAPK14ALDH1A1GAA
SCHEMBL955275 0.74 TAAR1 (0.66) TAAR1HTR1AADRA1AADRA2AADRA2B
SCHEMBL4627741 0.73 DPYD (0.36) AOC3MAPK14MAPK1NTSR1KDM4E
SCHEMBL953533 0.72 F2RL1 (0.39) MAPK14MAPK1ALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP claimed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO claimed