SCHEMBL4630440

SCHEMBL4630440

CN1CCN(CC(=O)C2CCCN2)CC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.42
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
DPP4 P27487 3/20 0.39
DPP8 Q6V1X1 2/20 0.39
DPP9 Q86TI2 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
FAP Q12884 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
PRCP P42785 1/20 0.37
KDM4E B2RXH2 1/20 0.36
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
NOS2 P35228 2/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Proline SCHEMBL28674176 0.76 DPP4 (0.46) DPP4DPP8DPP9FAPDPP7
SCHEMBL3832732 0.75 DPP4 (0.57) DPP4DPP8DPP9FAPDPP7
SCHEMBL3331935 0.75 DPP4 (0.57) DPP4DPP8DPP9FAPDPP7
Proline SCHEMBL28685641 0.75 DPP4 (0.45) DPP4DPP8DPP9FAPDPP7
SCHEMBL3331942 0.75 DPP4 (0.57) DPP4DPP8DPP9FAPDPP7
Proline SCHEMBL28688776 0.74 DPP4 (0.39) DPP4DPP8DPP9FAPDPP7
SCHEMBL878969 0.71
SCHEMBL805298 0.71
SCHEMBL14296418 0.71
SCHEMBL6202288 0.71 HTT (0.58) DPP4DPP8DPP9FAPDPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed