SCHEMBL4630575

SCHEMBL4630575

O=C(Oc1ccc(OC(F)(F)F)cc1)C1CCNC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.62
EPHX1 P07099 2/20 0.49
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
SSTR1 P30872 2/20 0.41
SSTR4 P31391 2/20 0.41
LIPE Q05469 1/20 0.40
EPHX2 P34913 3/20 0.40
SCN10A Q9Y5Y9 1/20 0.39
ELANE P08246 1/20 0.39
HSD11B1 P28845 1/20 0.39
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP13 P45452 1/20 0.39
MMP14 P50281 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15092031 0.83 HTT (0.61) HTR2CEPHX1HTTKMT2ASMN1; SMN2
SCHEMBL29175598 0.81 HTT (0.50) HTR2CHTTKMT2ASMN1; SMN2TDP1
SCHEMBL28061413 0.81 KMT2A (0.50) HTR2CHTTKMT2ASMN1; SMN2TDP1
SCHEMBL28167146 0.80 ELANE (0.51) HTTKMT2ASMN1; SMN2TDP1ELANE
SCHEMBL5813373 0.80 ELANE (0.51) HTTKMT2ASMN1; SMN2TDP1ELANE
SCHEMBL23390079 0.80 HTR2C (0.68) HTR2CEPHX1KMT2ASMN1; SMN2LIPE
SCHEMBL17488206 0.80 HTR2C (0.68) HTR2CEPHX1KMT2ASMN1; SMN2LIPE
SCHEMBL4630807 0.80 HTR2C (0.61) HTR2CEPHX1KMT2ASMN1; SMN2SSTR1
SCHEMBL27309277 0.79 KMT2A (0.66) EPHX1HTTKMT2ASMN1; SMN2TDP1
SCHEMBL23390539 0.78 HTR2C (0.56) HTR2CEPHX1TDP1SSTR1SSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed