SCHEMBL4633089

SCHEMBL4633089

OCCNCC(O)COCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.57
CA2 P00918 1/20 0.57
CA7 P43166 1/20 0.57
CA9 Q16790 1/20 0.57
CASR P41180 1/20 0.50
MAPK1 P28482 1/20 0.47
TSHR P16473 2/20 0.45
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
LMNA P02545 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.43
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4407591 1.00 CA1 (0.57) CA1CA2CA7CA9CASR
SCHEMBL30819084 0.86 CA1 (0.55) CA1CA2CA7CA9CASR
SCHEMBL30819056 0.86 CA1 (0.55) CA1CA2CA7CA9CASR
SCHEMBL30819079 0.86 CA1 (0.55) CA1CA2CA7CA9CASR
SCHEMBL11922728 0.86 CA1 (0.55) CA1CA2CA7CA9CASR
SCHEMBL31127313 0.86 CA1 (0.55) CA1CA2CA7CA9CASR
SCHEMBL24473808 0.84 CA1 (0.60) CA1CA2CA7CA9CASR
SCHEMBL17005403 0.84 CA1 (0.60) CA1CA2CA7CA9CASR
SCHEMBL2810250 0.84 CA1 (0.60) CA1CA2CA7CA9CASR
SCHEMBL24759135 0.79 ADRB1 (0.54) MAPK1TSHRKMT2AMEN1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924572-A1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SmithKline Beecham Corporation (US) 2008-05-28 EP disclosed
WO-2007030366-A1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed