SCHEMBL4634185

SCHEMBL4634185

COc1ccccc1OP(=O)(Cl)OC(=O)[C@H](C)NOCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
ACHE P22303 3/20 0.40
MMP2 P08253 1/20 0.39
CA9 Q16790 1/20 0.39
CASP3 P42574 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SMPD1 P17405 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.38
RXRA P19793 1/20 0.38
TP53 P04637 1/20 0.38
GLA P06280 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4634179 0.89 SMN1; SMN2 (0.39) NPC1RAB9ACA1CA2MMP2
SCHEMBL644062 0.88 NPC1 (0.51) NPC1RAB9ACA1CA2ACHE
SCHEMBL10004061 0.88 NPC1 (0.51) NPC1RAB9ACA1CA2ACHE
SCHEMBL857081 0.86 ELANE (0.48) NPC1RAB9ACA1CA2MMP2
SCHEMBL1027922 0.86 ALDH1A1 (0.40) NPC1RAB9ACA1CA2MMP2
SCHEMBL3977464 0.86 ALDH1A1 (0.40) NPC1RAB9ACA1CA2MMP2
SCHEMBL1807712 0.83 ELANE (0.42) NPC1RAB9ACA1CA2MMP2
SCHEMBL1808359 0.82 CA1 (0.50) NPC1RAB9ACA1CA2MMP2
SCHEMBL4277332 0.82 MEN1 (0.43) NPC1RAB9ACA1CA2MMP2
SCHEMBL4273425 0.82 CA1 (0.50) NPC1RAB9ACA1CA2MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928475-A2 ANTIVIRAL PHOSPHORAMIDATES OF 4'-SUBSTITUTED PRONUCLEOTIDES F.HOFFMANN-LA ROCHE AG (CH) 2008-06-11 EP disclosed
WO-2007020193-A2 ANTIVIRAL PHOSPHORAMIDATES OF 4 ' -SUBSTITUTED PRONUCLEOTIDES F. HOFFMANN-LA ROCHE AG (CH) 2007-02-22 WO disclosed