SCHEMBL4635655

SCHEMBL4635655

Cc1cccc(C#Cc2ccc3c(n2)CCCC3=O)c1.O=C1CCCc2nc(C#Cc3cccc(O)c3)ccc21.O=C1CCCc2nc(C#Cc3ccccc3)ccc21.O=C1CCCc2nc(C#Cc3cccnc3)ccc21

nearest known ligand 0.59

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 19/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4635256 0.86 GRM5 (0.49) GRM5
SCHEMBL4635014 0.86 GRM5 (0.81) GRM5
SCHEMBL4635073 0.83 GRM5 (0.42) GRM5
SCHEMBL4337210 0.83 GRM5 (0.71) GRM5
SCHEMBL4339145 0.83 GRM5 (0.71) GRM5
SCHEMBL4331723 0.82 GRM5 (0.73) GRM5
SCHEMBL4635784 0.78 GRM5 (0.37) GRM5
SCHEMBL4634745 0.78 GRM5 (0.53) GRM5
SCHEMBL4325876 0.77 GRM5 (1.00) GRM5
SCHEMBL4635572 0.75 GRM5 (0.48) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931635-A1 TETRAHYDROQUINOLINONES AND THEIR USE AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS Merz Pharma GmbH & Co.KGaA (DE) 2008-06-18 EP claimed
WO-2007023290-A1 TETRAHYDROQUINOLINONES AND THEIR USE AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERZ PHARMA GMBH & CO. KGAA (DE) 2007-03-01 WO claimed
EP-1931635-A1 TETRAHYDROQUINOLINONES AND THEIR USE AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS Merz Pharma GmbH & Co.KGaA (DE) 2008-06-18 EP disclosed
WO-2007023290-A1 TETRAHYDROQUINOLINONES AND THEIR USE AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERZ PHARMA GMBH & CO. KGAA (DE) 2007-03-01 WO disclosed