SCHEMBL4635903

SCHEMBL4635903

FC(F)(F)O[CH]Oc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
LTA4H P09960 1/20 0.36
ALDH1A1 P00352 1/20 0.33
CA4 P22748 1/20 0.33
PARP10 Q53GL7 1/20 0.32
MAOB P27338 1/20 0.32
PTPN1 P18031 1/20 0.31
KCNA3 P22001 1/20 0.31
CA5A P35218 2/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
PDK1 Q15118 1/20 0.30
PDK2 Q15119 1/20 0.30
PDK3 Q15120 1/20 0.30
PDK4 Q16654 1/20 0.30
GRIN2B Q13224 1/20 0.30
CA5B Q9Y2D0 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7658790 0.80 TSHR (0.35) TSHRLTA4HALDH1A1CA4MAOB
SCHEMBL712888 0.77 CA4 (0.39) TSHRLTA4HALDH1A1CA4KCNA3
SCHEMBL6606014 0.77 LTA4H (0.50) TSHRLTA4HALDH1A1CA4PARP10
SCHEMBL28369275 0.75 LTA4H (0.47) TSHRLTA4HALDH1A1CA4PARP10
SCHEMBL3630500 0.71 LTA4H (0.39) TSHRLTA4HALDH1A1CA4MAOB
SCHEMBL1543834 0.69 CA4 (0.50) TSHRLTA4HCA4MAOBKCNA3
SCHEMBL20869702 0.68 TSHR (0.36) TSHRLTA4HALDH1A1CA4MAOB
SCHEMBL20856386 0.68 TSHR (0.36) TSHRLTA4HALDH1A1CA4MAOB
SCHEMBL20856387 0.68 TSHR (0.36) TSHRLTA4HALDH1A1CA4MAOB
SCHEMBL196320 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102895230-A Antituberculous composition comprising oxazole compounds OTSUKA PHARMA CO LTD 2013-01-30 CN disclosed
CN-101277740-B Antituberculous composition comprising azole compound OTSUKA PHARMA CO LTD 2012-12-05 CN disclosed
CN-101277740-A Antituberculous compositions comprising * azole compounds OTSUKA PHARMA CO LTD (JP) 2008-10-01 CN disclosed
EP-1931425-A1 ANTITUBERCULOUS COMPOSITION COMPRISING OXAZOLE COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-06-18 EP disclosed
WO-2007043542-A1 ANTITUBERCULOUS COMPOSITION COMPRISING OXAZOLE COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-04-19 WO disclosed