SCHEMBL4635985

SCHEMBL4635985

N#CCCNCCc1ccc(Cl)c(Cl)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.63
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
PNMT P11086 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
ROCK1 Q13464 1/20 0.42
PYGL P06737 1/20 0.41
NR1I3 Q14994 1/20 0.41
IDO1 P14902 1/20 0.40
HTR1A P08908 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
HTR2A P28223 1/20 0.40
HTR7 P34969 1/20 0.40
HTR2B P41595 1/20 0.40
HTR5A P47898 1/20 0.40
IGF1R P08069 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637177 0.90 SIGMAR1 (0.55) SIGMAR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL14846267 0.79 IGF1R (0.53) SIGMAR1CYP1A2CYP2C19PNMTTAAR1
SCHEMBL17186234 0.77 SIGMAR1 (0.54) SIGMAR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL11279010 0.77 SIGMAR1 (0.69) SIGMAR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL14829408 0.77 IGF1R (0.56) SIGMAR1CYP1A2CYP2C19PNMTTAAR1
SCHEMBL17055956 0.77 DRD1 (0.56) SIGMAR1CYP1A2CYP2D6TAAR1HTR1A
SCHEMBL12168011 0.75 SIGMAR1 (0.66) SIGMAR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL14149435 0.75 SIGMAR1 (0.70) SIGMAR1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL11739917 0.74 ATM (0.61) SIGMAR1ALOX15
SCHEMBL2850382 0.73 SIGMAR1 (0.59) SIGMAR1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931620-A1 AMINO-ALKYL-AMIDE DERIVATIVES AS CCR3 RECEPTOR LIQUIDS Sanofi-Aventis (FR) 2008-06-18 EP disclosed
WO-2007034252-A1 AMINO-ALKYL-AMIDE DERIVATIVES AS CCR3 RECEPTOR LIQUIDS SANOFI-AVENTIS (FR) 2007-03-29 WO disclosed