SCHEMBL4636772

SCHEMBL4636772

CC#CCn1c(=O)[nH]c(=O)c2c1nc(C#Cc1cccc(OCCOC)c1)n2C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
KMT2A Q03164 6/20 0.42
HPGD P15428 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
XBP1 P17861 1/20 0.42
MAPK1 P28482 3/20 0.40
LMNA P02545 2/20 0.40
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 2/20 0.37
TP53 P04637 2/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PKM P14618 1/20 0.37
MEN1 O00255 3/20 0.36
ATM Q13315 1/20 0.36
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
MPO P05164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637377 0.79 HPGD (0.40) ALDH1A1KMT2AHPGDNPSR1XBP1
SCHEMBL2542698 0.77 ADORA1 (0.47) ALDH1A1LMNASMN1; SMN2HTT
SCHEMBL2537017 0.69 KDM4E (0.47) ALDH1A1KMT2AHPGDNPSR1XBP1
SCHEMBL4950417 0.68 ADORA1 (0.53)
SCHEMBL2537641 0.68 ADORA2A (0.46)
SCHEMBL16199473 0.68 MAPT (0.44) ALDH1A1KMT2AHPGDNPSR1XBP1
SCHEMBL2541481 0.67 ADORA2A (0.49)
SCHEMBL2535874 0.67 ADORA1 (0.45)
SCHEMBL2537944 0.66 ADORA1 (0.44)
SCHEMBL2536366 0.66 ADORA1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed