SCHEMBL4637046

SCHEMBL4637046

Cc1ccccc1C(I)N=C=O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
ACP3 P15309 1/20 0.36
TSHR P16473 1/20 0.33
ACHE P22303 1/20 0.33
ALDH1A1 P00352 2/20 0.32
CYP3A4 P08684 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
GAA P10253 1/20 0.31
MEN1 O00255 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL163750 0.80 ESR1 (0.43) ESR1ACP3TSHRACHEALDH1A1
SCHEMBL8755636 0.78 ESR1 (0.42) ESR1ACP3TSHRACHEALDH1A1
SCHEMBL27978287 0.78 ESR1 (0.42) ESR1ACP3TSHRACHEALDH1A1
SCHEMBL4455459 0.72 ACP3 (0.39) ESR1ACP3ALDH1A1GAAMEN1
SCHEMBL10902580 0.70 ESR1 (0.34) ESR1ACP3TSHRACHEALDH1A1
SCHEMBL23361811 0.69 ESR1 (0.54) ESR1ACP3TSHRACHEALDH1A1
SCHEMBL27510474 0.69 CYP3A4 (0.39) ESR1TSHRCYP3A4SLC6A2MAPT
SCHEMBL331134 0.69 MIF (0.39) TSHRALDH1A1CYP3A4SLC6A2LMNA
SCHEMBL7331227 0.68 ESR1 (0.52) ESR1ACP3TSHRACHEALDH1A1
SCHEMBL3981386 0.68 ESR1 (0.31) ESR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893590-A1 BENZOOXAZOLE-2-ON DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS Sanofi-Aventis (FR) 2008-03-05 EP disclosed
EP-1874741-A1 AZOLE DERIVATIVES IN THE FORM OF LIPASE AND PHOSPHOLIPASE INHIBITORS sanofi-aventis (FR) 2008-01-09 EP disclosed
WO-2006131233-A1 BENZOOXAZOLE-2-ON DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS SANOFI-AVENTIS (FR) 2006-12-14 WO disclosed
WO-2006111321-A1 AZOLE DERIVATIVES IN THE FORM OF LIPASE AND PHOSPHOLIPASE INHIBITORS SANOFI-AVENTIS (DE) 2006-10-26 WO disclosed