SCHEMBL4637977

SCHEMBL4637977

O=C(c1ncn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1)c1c(COC2CCCCO2)noc1-c1ccccc1Cl

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 10/20 0.34
S1PR5 Q9H228 3/20 0.34
S1PR4 O95977 2/20 0.34
RORC P51449 2/20 0.33
TACR1 P25103 3/20 0.33
PPARD Q03181 1/20 0.32
S1PR3 Q99500 6/20 0.32
KCNH2 Q12809 2/20 0.32
CFTR P13569 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C8 P10632 1/20 0.31
SCD5 Q86SK9 1/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637899 0.94 IDH1 (0.32) S1PR1S1PR5S1PR4RORCTACR1
SCHEMBL4639054 0.88 ALDH1A1 (0.36) S1PR1S1PR5S1PR4RORCTACR1
SCHEMBL4637919 0.85 TACR1 (0.37) S1PR1S1PR5S1PR4TACR1PPARD
SCHEMBL4638821 0.84 TACR1 (0.32) RORCTACR1CFTRCYP3A4POLB
SCHEMBL4638616 0.84 CFTR (0.33) S1PR1S1PR5S1PR4RORCTACR1
SCHEMBL4638809 0.83 ALDH1A1 (0.36) S1PR1S1PR5S1PR4RORCPPARD
SCHEMBL4637728 0.83 IDH1 (0.37) RORCTACR1CFTR
SCHEMBL4637808 0.81 TACR1 (0.39) TACR1CYP3A4
SCHEMBL4639496 0.81 CFTR (0.32) CFTRCYP3A4
SCHEMBL4637743 0.80 IDH1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed