SCHEMBL4638012

SCHEMBL4638012

Cc1c(C(=O)O)ccc(-c2cc[n+]([O-])cc2)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
NR4A1 P22736 1/20 0.33
RECQL P46063 1/20 0.33
ESR2 Q92731 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP1A2 P05177 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SLC22A6 Q4U2R8 1/20 0.32
SLC22A8 Q8TCC7 1/20 0.32
RAB9A P51151 1/20 0.32
HAAO P46952 1/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974190 0.80 ALDH1A1 (0.49) SMN1; SMN2MEN1KMT2AALDH1A1RAB9A
SCHEMBL843489 0.78 CYP1A2 (0.48) TSHRHSD17B10SMN1; SMN2MEN1KMT2A
SCHEMBL842987 0.77 FOLH1 (0.49) TSHRHSD17B10SMN1; SMN2ALDH1A1RAB9A
SCHEMBL27547124 0.76 KDM4E (0.43) HSD17B10SMN1; SMN2MEN1KMT2APOLB
SCHEMBL4140940 0.74 CA9 (0.51)
SCHEMBL128319 0.73 CYP1A2 (0.58) TSHRHSD17B10SMN1; SMN2MEN1KMT2A
SCHEMBL31389208 0.73 CYP1A2 (0.58) TSHRHSD17B10SMN1; SMN2MEN1KMT2A
SCHEMBL28503156 0.71 EGFR (0.52) TSHRHSD17B10SMN1; SMN2MEN1KMT2A
Ammonia Solution, Strong SCHEMBL29137499 0.71 CYP1A2 (0.55) TSHRHSD17B10SMN1; SMN2MEN1KMT2A
Ethylene Glycol SCHEMBL25205438 0.69 CYP1A2 (0.48) TSHRHSD17B10MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951708-A2 PIPERAZINE DERIVATIVES USEFUL AS CCR5 ANTAGONISTS SCHERING CORPORATION (US) 2008-08-06 EP disclosed
WO-2007050375-A2 PIPERAZINE DERIVATIVES USEFUL AS CCR5 ANTAGONISTS SCHERING CORPORATION (US) 2007-05-03 WO disclosed