SCHEMBL4638508

SCHEMBL4638508

O=C(C#Cc1ccccc1Cl)c1nnn(Cc2cc(Cl)cc(Cl)c2)c1-c1ccncc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.42
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 1/20 0.38
P2RX7 Q99572 1/20 0.36
HPGD P15428 1/20 0.34
IDO1 P14902 2/20 0.34
TDO2 P48775 1/20 0.34
GALR3 O60755 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
NR2F2 P24468 1/20 0.34
HIF1A Q16665 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638811 0.90 IDH1 (0.40) CYP19A1ALDH1A1TSHRSMN1; SMN2MAPT
SCHEMBL4637813 0.88 IDH1 (0.39) CYP19A1ALDH1A1TSHRSMN1; SMN2CYP3A4
SCHEMBL4638053 0.81 ALDH1A1 (0.44) CYP19A1ALDH1A1TSHRMAPTPOLB
SCHEMBL4638504 0.81 CYP19A1 (0.36) CYP19A1ALDH1A1TSHRSMN1; SMN2MAPT
SCHEMBL4638905 0.79 IDH1 (0.41) CYP19A1ALDH1A1TSHRSMN1; SMN2MAPT
SCHEMBL4637714 0.79 IDH1 (0.54) CYP19A1ALDH1A1TSHRP2RX7HIF1A
SCHEMBL4639451 0.79 CYP19A1 (0.48) CYP19A1ALDH1A1TSHRSMN1; SMN2P2RX7
SCHEMBL4707915 0.79 IDH1 (0.48) CYP19A1ALDH1A1TSHRP2RX7
SCHEMBL4637949 0.78 IDH1 (0.39) CYP19A1ALDH1A1TSHRSMN1; SMN2MAPT
SCHEMBL4707175 0.77 MAPT (0.46) ALDH1A1TSHRSMN1; SMN2MAPTP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed