Sulfamide

Sulfamide

SCHEMBL4638912

Cc1onc(-c2ccccc2)c1-c1ccccc1.NS(N)(=O)=O

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.81
PTGS1 P23219 9/20 0.81
MT-CO2 P00403 3/20 0.81
CA12 O43570 1/20 0.81
CA1 P00915 1/20 0.81
CA2 P00918 1/20 0.81
LMNA P02545 1/20 0.81
CA3 P07451 1/20 0.81
ADRB2 P07550 1/20 0.81
ADRB1 P08588 1/20 0.81
CYP3A4 P08684 1/20 0.81
ADORA3 P0DMS8 1/20 0.81
CHRM1 P11229 1/20 0.81
ADRA2B P18089 1/20 0.81
CA4 P22748 1/20 0.81
CA6 P23280 1/20 0.81
SLC6A2 P23975 1/20 0.81
PDE4A P27815 1/20 0.81
ADORA1 P30542 1/20 0.81
CA5A P35218 1/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6245202 0.90 PTGS2 (0.80) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL6168344 0.90 PTGS2 (1.00) PTGS2PTGS1MT-CO2CA12CA1
Valdecoxib SCHEMBL3356 0.90 PTGS2 (1.00) PTGS2PTGS1MT-CO2CA12CA1
Valdecoxib SCHEMBL3853130 0.90 PTGS2 (1.00) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL2277199 0.89 PTGS2 (1.00) PTGS2PTGS1MT-CO2CA12CA1
Sulfuric Acid SCHEMBL6263326 0.89 PTGS2 (0.77) PTGS2PTGS1MT-CO2CA12CA1
Sulfuric Acid SCHEMBL6263325 0.89 PTGS2 (0.77) PTGS2PTGS1MT-CO2CA12CA1
Valdecoxib SCHEMBL6601157 0.88 PTGS2 (0.97) PTGS2PTGS1MT-CO2CA12CA1
Valdecoxib SCHEMBL5999213 0.88 PTGS2 (0.97) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL28961699 0.86 PTGS2 (0.79) PTGS2PTGS1MT-CO2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1479385-B1 Use of cyclooxygenase-2 inhibitors in the treatment and prevention of neoplasia SEARLE LLC (US) 2008-07-02 EP claimed
WO-2005085218-A1 A NOVEL PROCESS FOR PREPARING VALDECOXIB THAKASHINAMOORTHY CHANDIRAN (IN) 2005-09-15 WO disclosed