SCHEMBL4639581

SCHEMBL4639581

O=C(N[C@H]1CCCC1=O)OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
GAA P10253 1/20 0.56
TSHR P16473 1/20 0.53
EPHX1 P07099 1/20 0.53
NAAA Q02083 3/20 0.53
TLR4 O00206 1/20 0.53
CTSK P43235 2/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
ASAH1 Q13510 1/20 0.48
CPB1 P15086 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18029925 1.00 ALDH1A1 (0.56) ALDH1A1GAATSHREPHX1NAAA
SCHEMBL760401 0.96 EPHX1 (0.59) ALDH1A1GAATSHREPHX1NAAA
SCHEMBL14534711 0.96 EPHX1 (0.59) ALDH1A1GAATSHREPHX1NAAA
SCHEMBL425375 0.92 ALDH1A1 (0.58) ALDH1A1GAATSHREPHX1NAAA
SCHEMBL1987472 0.84 ALDH1A1 (0.53) ALDH1A1GAATSHREPHX1NAAA
SCHEMBL20178484 0.84 ALDH1A1 (0.53) ALDH1A1GAATSHREPHX1NAAA
SCHEMBL12640899 0.84 ALDH1A1 (0.53) ALDH1A1GAATSHREPHX1NAAA
SCHEMBL12564549 0.84 ALDH1A1 (0.53) ALDH1A1GAATSHREPHX1NAAA
SCHEMBL1987474 0.84 ALDH1A1 (0.53) ALDH1A1GAATSHREPHX1NAAA
SCHEMBL1718075 0.83 TLR4 (0.56) ALDH1A1GAATSHREPHX1NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954668-A2 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS Brystol-Myers Squibb Company (US) 2008-08-13 EP disclosed
EP-1951673-A2 HETEROCYCLIC CETP INHIBITORS Bristol-Myers Squibb Company (US) 2008-08-06 EP disclosed
WO-2007062314-A2 HETEROCYCLIC CETP INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-31 WO disclosed
WO-2007062308-A2 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-31 WO disclosed