Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL4639804

CC(C)(CCn1cnc2cc(Cl)c(OC(=O)O)cc21)NC[C@H](O)c1cccc(NS(=O)(=O)c2ccccc2)c1.O=C(O)C(F)(F)F

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 7/20 0.41
NR1I2 O75469 7/20 0.37
HPGD P15428 2/20 0.36
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
HTR6 P50406 1/20 0.35
ALDH1A1 P00352 2/20 0.34
CBLB Q13191 1/20 0.34
ADRA1A P35348 2/20 0.34
MEN1 O00255 1/20 0.34
PKM P14618 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4642662 0.97 ADRB3 (0.41) ADRB3NR1I2HPGDADRB2ADRB1
SCHEMBL4640331 0.97 ADRB3 (0.41) ADRB3NR1I2HPGDADRB2ADRB1
SCHEMBL4648541 0.94 ADRB3 (0.41) ADRB3NR1I2HPGDADRB2ADRB1
SCHEMBL4645527 0.94 ADRB3 (0.41) ADRB3NR1I2HPGDADRB2ADRB1
Trifluoroacetic Acid SCHEMBL4605859 0.93 ADRB3 (0.42) ADRB3NR1I2HPGDHTR6ALDH1A1
Trifluoroacetic Acid SCHEMBL4646187 0.92 ADRB3 (0.41) ADRB3NR1I2HPGDADRB2ADRB1
Trifluoroacetic Acid SCHEMBL4642328 0.91 ADRB3 (0.41) ADRB3NR1I2HPGDADRB2ADRB1
Trifluoroacetic Acid SCHEMBL4916366 0.90 ADRB3 (0.41) ADRB3NR1I2HPGDHTR6ALDH1A1
Trifluoroacetic Acid SCHEMBL4642020 0.89 ADRB3 (0.41) ADRB3NR1I2HPGDADRB2ADRB1
Trifluoroacetic Acid SCHEMBL4913411 0.89 ADRB3 (0.41) ADRB3NR1I2HPGDHTR6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed