SCHEMBL4639963

SCHEMBL4639963

COC(=O)Oc1ccc2c(c1)[nH]c(=O)n2CCC(C)(C)NCC(O)c1cccc(NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 15/20 0.42
ADRB2 P07550 2/20 0.38
ADRB1 P08588 1/20 0.38
ADRA1A P35348 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4647049 0.92 ADRB3 (0.42) ADRB3ADRB2ADRB1ADRA1A
SCHEMBL4918038 0.89 ADRB3 (0.41) ADRB3ADRB2ADRB1ALDH1A1PKM
SCHEMBL14185303 0.88 ADRB3 (0.42) ADRB3ADRB2ADRB1
SCHEMBL4606960 0.88 ADRB3 (0.45) ADRB3ADRB2ADRB1
Trifluoroacetic Acid SCHEMBL4642656 0.85 ADRB3 (0.40) ADRB3ADRB2ADRB1
SCHEMBL4918874 0.84 ADRB3 (0.38) ADRB3ADRB2ADRB1ADRA1A
SCHEMBL4642663 0.84 ADRB3 (0.37) ADRB3ALDH1A1PKMTSHRMAPK1
SCHEMBL4637273 0.83 ADRB3 (0.42) ADRB3ADRB2ADRB1
SCHEMBL4639973 0.83 ADRB3 (0.42) ADRB3ADRB2ADRB1
Trifluoroacetic Acid SCHEMBL4639441 0.80 ADRB3 (0.41) ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed