SCHEMBL4642663

SCHEMBL4642663

CC(C)(CCn1c(=O)[nH]c2cc(OC(=O)O)ccc21)NCC(OC(=O)C(F)(F)F)c1cccc(NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 2/20 0.37
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
DUT P33316 1/20 0.33
SERPINE1 P05121 1/20 0.33
BRAF P15056 3/20 0.32
ALDH1A1 P00352 1/20 0.32
PKM P14618 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
MAPT P10636 4/20 0.32
TP53 P04637 2/20 0.32
KMT2A Q03164 1/20 0.32
FABP4 P15090 1/20 0.32
EPHX2 P34913 1/20 0.31
PPARG P37231 1/20 0.31
TRIM24 O15164 1/20 0.31
POLB P06746 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4918872 0.91 MEN1 (0.37) ADRB3OPRM1OPRD1MAPTKMT2A
Trifluoroacetic Acid SCHEMBL4647049 0.89 ADRB3 (0.42) ADRB3SERPINE1
SCHEMBL4639786 0.84 ADRB3 (0.42) ADRB3OPRM1OPRD1ALDH1A1PKM
SCHEMBL4639963 0.84 ADRB3 (0.42) ADRB3ALDH1A1PKMTSHRMAPK1
SCHEMBL4645777 0.83 ADRB3 (0.40) ADRB3OPRM1OPRD1ALDH1A1PKM
SCHEMBL4918874 0.81 ADRB3 (0.38) ADRB3SERPINE1MAPTEPHX2PPARG
Trifluoroacetic Acid SCHEMBL4642656 0.79 ADRB3 (0.40) ADRB3SERPINE1MAPTKMT2AEPHX2
SCHEMBL4605628 0.78 ADRB3 (0.42) ADRB3OPRM1OPRD1ALDH1A1PKM
SCHEMBL4830639 0.78 ADRB3 (0.36) ADRB3OPRM1OPRD1ALDH1A1PKM
SCHEMBL4639769 0.78 ADRB3 (0.36) ADRB3OPRM1OPRD1ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed