SCHEMBL4642404

SCHEMBL4642404

COc1cc2c(cc1OC(=O)O)ncn2CCC(C)(C)NC[C@H](O)c1cccc(NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 12/20 0.41
HPGD P15428 4/20 0.41
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 1/20 0.41
PKM P14618 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
LRRK2 Q5S007 1/20 0.39
NR1I2 O75469 1/20 0.38
LMNA P02545 2/20 0.38
MAPT P10636 2/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ALOX12 P18054 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4641939 1.00 ADRB3 (0.41) ADRB3HPGDALDH1A1MEN1PKM
Trifluoroacetic Acid SCHEMBL4646187 0.97 ADRB3 (0.41) ADRB3HPGDALDH1A1MEN1PKM
SCHEMBL4649033 0.92 ADRB3 (0.42) ADRB3HPGDALDH1A1MEN1PKM
SCHEMBL4649135 0.92 ADRB3 (0.42) ADRB3HPGDALDH1A1MEN1PKM
SCHEMBL4642662 0.92 ADRB3 (0.41) ADRB3HPGDALDH1A1MEN1PKM
SCHEMBL4648541 0.92 ADRB3 (0.41) ADRB3HPGDALDH1A1MEN1PKM
SCHEMBL4645527 0.92 ADRB3 (0.41) ADRB3HPGDALDH1A1MEN1PKM
SCHEMBL4640331 0.92 ADRB3 (0.41) ADRB3HPGDALDH1A1MEN1PKM
SCHEMBL4641932 0.91 ADRB3 (0.42) ADRB3HPGDALDH1A1MEN1PKM
SCHEMBL4916291 0.91 ADRB3 (0.42) ADRB3HPGDALDH1A1MEN1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP claimed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO claimed
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed