SCHEMBL4643542

SCHEMBL4643542

CC1(C)CCCCC2(CC(c3ccccc3)=NO2)CC(C)(C)C1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.55
CHRNA3 P32297 1/20 0.55
NLRP3 Q96P20 1/20 0.38
RECQL P46063 1/20 0.38
SSTR5 P35346 1/20 0.35
POLB P06746 1/20 0.34
CYP2C9 P11712 4/20 0.33
KCNH2 Q12809 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2205534 0.88 CHRNB4 (0.52) CHRNB4CHRNA3NLRP3RECQLSSTR5
SCHEMBL4643127 0.84 CHRNB4 (0.40) CHRNB4CHRNA3CYP2C9KCNH2
SCHEMBL10210780 0.72 CHRNB4 (0.55) CHRNB4CHRNA3NLRP3RECQLSSTR5
SCHEMBL2210658 0.71 CHRNB4 (0.36) CHRNB4CHRNA3NLRP3RECQLTDP1
SCHEMBL5015649 0.71 CHRNB4 (0.54) CHRNB4CHRNA3NLRP3RECQLCYP2C9
SCHEMBL895210 0.71 CHRNB4 (0.54) CHRNB4CHRNA3NLRP3RECQLSSTR5
SCHEMBL14534188 0.71 CHRNB4 (0.53) CHRNB4CHRNA3NLRP3RECQLSSTR5
Ammonia Solution, Strong SCHEMBL5126795 0.70 CHRNB4 (0.53) CHRNB4CHRNA3NLRP3RECQLCYP2C9
SCHEMBL5015653 0.70 CHRNB4 (0.52) CHRNB4CHRNA3NLRP3RECQLSSTR5
SCHEMBL10168605 0.69 CHRNB4 (0.52) CHRNB4CHRNA3NLRP3RECQLSSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888542-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2008-02-20 EP claimed
WO-2006136245-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2006-12-28 WO claimed
EP-1888542-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2008-02-20 EP disclosed
WO-2006136245-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2006-12-28 WO disclosed