SCHEMBL4646374

SCHEMBL4646374

O=C1CN(c2cc(Br)ccc2O)S(=O)(=O)N1

nearest known ligand 0.60

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 12/20 0.60
PTPN2 P17706 13/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL629685 0.85 PTPN1 (0.70) PTPN1PTPN2
SCHEMBL3223697 0.82 PTPN1 (0.60) PTPN1PTPN2
SCHEMBL6685010 0.79 PTPN1 (0.67) PTPN1PTPN2
SCHEMBL2934032 0.79 PTPN1 (0.70) PTPN1PTPN2
SCHEMBL2937132 0.79 PTPN1 (0.77) PTPN1PTPN2
SCHEMBL3921154 0.79 PTPN1 (0.59) PTPN1PTPN2
SCHEMBL12056226 0.78 PTPN1 (0.60) PTPN1PTPN2
SCHEMBL2935490 0.78 PTPN1 (0.65) PTPN1PTPN2
SCHEMBL2936747 0.78 PTPN1 (0.65) PTPN1PTPN2
SCHEMBL6687346 0.78 PTPN1 (0.66) PTPN1PTPN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080293782-A1 1,1,3-Trioxo-1,2,5-Thiadiazolidines and Their Use as Ptp-Ases Inhibitors NOVARTIS AG (CH) 2008-11-27 US disclosed
EP-1960377-A1 l , l , 3-TRI0X0-l , 2 , 5-THIADIAZ0LIDINES AND THEIR USE AS PTP-ASES INHIBITORS Novartis AG (CH) 2008-08-27 EP disclosed
WO-2007067614-A1 l, l, 3-TRI0X0-l, 2, 5-THIADIAZ0LIDINES AND THEIR USE AS PTP-ASES INHIBITORS NOVARTIS AG (CH) 2007-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080293782-A1 1,1,3-Trioxo-1,2,5-Thiadiazolidines and Their Use as Ptp-Ases Inhibitors PTPRS, IRS1, PTPMT1 PTPN1 10/4885PTPN2 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.